Chemistry:Desmethylmoramide

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Short description: Opioid analgesic drug
Desmethylmoramide
Desmethylmoramide.svg
Names
Preferred IUPAC name
4-(Morpholin-4-yl)-2,2-diphenyl-1-(pyrrolidin-1-yl)butan-1-one
Identifiers
3D model (JSmol)
ChEMBL
ChemSpider
UNII
Properties
C24H30N2O2
Molar mass 378.516 g·mol−1
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
Infobox references
Tracking categories (test):

Desmethylmoramide (INN) is an opioid analgesic related to dextromoramide (the active (+)-isomer of moramide) that was synthesized and characterized in the late 1950s but was never marketed.[1][2][3]

See also

References

  1. The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. 14 November 2014. pp. 363–. ISBN 978-1-4757-2085-3. https://books.google.com/books?id=0vXTBwAAQBAJ&pg=PA363. 
  2. Concise Dictionary of Pharmacological Agents: Properties and Synonyms. Springer Science & Business Media. 6 December 2012. pp. 94–. ISBN 978-94-011-4439-1. https://books.google.com/books?id=tsjrCAAAQBAJ&pg=PA94. 
  3. "A new series of potent analgesics: dextro 2:2-diphenyl-3-methyl-4-morpholino-butyrylpyrrolidine and related amides. I. Chemical structure and pharmacological activity". The Journal of Pharmacy and Pharmacology 9 (6): 381–400. June 1957. doi:10.1111/j.2042-7158.1957.tb12290.x. PMID 13439527. 

Further reading

  • "New Psychotropic Agents. V. Derivatives of 5-Cyano- and 5-Carboxamidodibenzo[a,d]cycloheptadiene". Journal of Medicinal Chemistry 6 (3): 251–255. May 1963. doi:10.1021/jm00339a008. PMID 14185978.